| Tag |
Content |
LipidDB ID |
LipidDB-9606-00684 |
Entry Name |
|
UniProt Accession |
|
Theoretical PI |
6.42 |
Molecular Weight |
34655.91 |
Genbank Protein ID |
|
Genbank Nucleotide ID |
|
Protein Name |
Serine/threonine-protein kinase 16 |
Protein Synonyms/Alias |
2.7.11.1; Myristoylated and palmitoylated serine/threonine-protein kinase; MPSK; Protein kinase PKL12; TGF-beta-stimulated factor 1; TSF-1; Tyrosine-protein kinase STK16; 2.7.10.2; hPSK; |
Gene Name |
STK16 |
Gene Synonyms/Alias |
MPSK1; PKL12; TSF1; |
Created Date |
21-FEB-2001 |
| Lipid Modification Sites |
| Position |
Sequence Form |
Peptide |
References |
Modification Type |
2 | Canonical | ******MGHALCVCS | [1] | N-Myristoylation |
|
Organism |
Homo sapiens (Human) |
NCBI Taxa ID |
9606 |
Reference |
[1] Berson AE, Young C, Morrison SL, Fujii GH, Sheung J, Wu B, Bolen JB, BurkhardtAL. Identification and characterization of a myristylated and palmitylatedserine/threonine protein kinase. Biochem Biophys Res Commun. 1999 Jun16;259(3):533-8.[ PMID:10364453]
|
Functional Description |
Membrane-associated protein kinase that phosphorylates on serine and threonine residues. In vitro substrates include DRG1, ENO1 and EIF4EBP1. Also autophosphorylates. May be involved in secretory vesicle trafficking or intracellular signaling. May have a role in regulating stromal-epithelial interactions that occur during ductal morphogenesis in the mammary gland. May be involved in TGF-beta signaling. Able to autophosphorylate on Tyr residue; it is however unclear whether it has tyrosine-protein kinase toward other proteins. |
Sequence Annotation |
Domain: 20 293 Protein kinase. Nucleotide-binding: 26 34 ATP. Region: 166 202 Activation loop. Active site: 148 148 Proton acceptor. Binding site: 49 49 ATP. Modified residue: 185 185 Phosphothreonine; by autocatalysis. Modified residue: 197 197 Phosphoserine; by autocatalysis. Modified residue: 198 198 Phosphotyrosine; by autocatalysis.
|
Protein Length |
305 AA. |
Protein Sequence (Canonical) |
MGHALCVCSR GTVIIDNKRY LFIQKLGEGG FSYVDLVEGL HDGHFYALKR ILCHEQQDRE 60
EAQREADMHR LFNHPNILRL VAYCLRERGA KHEAWLLLPF FKRGTLWNEI ERLKDKGNFL 120
TEDQILWLLL GICRGLEAIH AKGYAHRDLK PTNILLGDEG QPVLMDLGSM NQACIHVEGS 180
RQALTLQDWA AQRCTISYRA PELFSVQSHC VIDERTDVWS LGCVLYAMMF GEGPYDMVFQ 240
KGDSVALAVQ NQLSIPQSPR HSSALRQLLN SMMTVDPHQR PHIPLLLSQL EALQPPAPGQ 300
HTTQI 305
|
FASTA (Canonical) |
>LipidDB-9606-00684|O75716
MGHALCVCSRGTVIIDNKRYLFIQKLGEGGFSYVDLVEGLHDGHFYALKRILCHEQQDRE
EAQREADMHRLFNHPNILRLVAYCLRERGAKHEAWLLLPFFKRGTLWNEIERLKDKGNFL
TEDQILWLLLGICRGLEAIHAKGYAHRDLKPTNILLGDEGQPVLMDLGSMNQACIHVEGS
RQALTLQDWAAQRCTISYRAPELFSVQSHCVIDERTDVWSLGCVLYAMMFGEGPYDMVFQ
KGDSVALAVQNQLSIPQSPRHSSALRQLLNSMMTVDPHQRPHIPLLLSQLEALQPPAPGQ
HTTQI
|
Gene Ontology |
GO:0005798; C:Golgi-associated vesicle; IEA:Ensembl GO:0016020; C:membrane; IEA:UniProtKB-KW GO:0005524; F:ATP binding; IEA:UniProtKB-KW GO:0004715; F:non-membrane spanning protein tyrosine kinase activity; IEA:UniProtKB-EC GO:0004674; F:protein serine/threonine kinase activity; IEA:UniProtKB-KW GO:0001077; F:RNA polymerase II core promoter proximal region sequence-specific DNA binding transcription factor activity involved in positive regulation of transcription; IEA:Ensembl GO:0071560; P:cellular response to transforming growth factor beta stimulus; IEA:Ensembl GO:0046777; P:protein autophosphorylation; IDA:UniProtKB |
Interpro |
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Pfam |
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SMART |
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PROSITE |
PROSITE; PS50011; PROTEIN_KINASE_DOM; PROSITE; PS00108; PROTEIN_KINASE_ST; |
PRINTS |
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